Dyclone
Dyclone Brand names, Dyclone Analogs
Dyclone Brand Names Mixture
- No information avaliable
Dyclone Chemical_Formula
C22H26N2O2S
Dyclone RX_link
http://www.rxlist.com/cgi/generic3/relpax.htm
Dyclone fda sheet
Dyclone msds (material safety sheet)
Dyclone Synthesis Reference
No information avaliable
Dyclone Molecular Weight
382.52 g/mol
Dyclone Melting Point
No information avaliable
Dyclone H2O Solubility
Readily soluble as hydrobromide formulation
Dyclone State
Solid
Dyclone LogP
3.587
Dyclone Dosage Forms
Tablet for oral administration (24.2 or 48.5 mg)
Dyclone Indication
For the acute treatment of migraine with or without aura in adults.
Dyclone Pharmacology
Eletriptan is a selective 5-hydroxytryptamine 1B/1D receptor agonist. In the anesthetized dog, eletriptan has been shown to reduce carotid arterial blood flow, with only a small increase in arterial blood pressure at high doses. While the effect on blood flow was selective for the carotid arterial bed, decreases in coronary artery diameter were observed. Eletriptan has also been shown to inhibit trigeminal nerve activity in the rat.
Dyclone Absorption
Well absorbed after oral administration with a mean absolute bioavailability of approximately 50%.
Dyclone side effects and Toxicity
Based on the pharmacology of the 5-HT1B/1D agonists, hypertension or other more serious cardiovascular symptoms could occur on overdose.
Dyclone Patient Information
No information avaliable
Dyclone Organisms Affected
Humans and other mammals
