Dyclocaine
Dyclocaine Brand names, Dyclocaine Analogs
Dyclocaine Brand Names Mixture
- No information avaliable
Dyclocaine Chemical_Formula
C22H26N2O2S
Dyclocaine RX_link
http://www.rxlist.com/cgi/generic3/relpax.htm
Dyclocaine fda sheet
Dyclocaine msds (material safety sheet)
Dyclocaine Synthesis Reference
No information avaliable
Dyclocaine Molecular Weight
382.52 g/mol
Dyclocaine Melting Point
No information avaliable
Dyclocaine H2O Solubility
Readily soluble as hydrobromide formulation
Dyclocaine State
Solid
Dyclocaine LogP
3.587
Dyclocaine Dosage Forms
Tablet for oral administration (24.2 or 48.5 mg)
Dyclocaine Indication
For the acute treatment of migraine with or without aura in adults.
Dyclocaine Pharmacology
Eletriptan is a selective 5-hydroxytryptamine 1B/1D receptor agonist. In the anesthetized dog, eletriptan has been shown to reduce carotid arterial blood flow, with only a small increase in arterial blood pressure at high doses. While the effect on blood flow was selective for the carotid arterial bed, decreases in coronary artery diameter were observed. Eletriptan has also been shown to inhibit trigeminal nerve activity in the rat.
Dyclocaine Absorption
Well absorbed after oral administration with a mean absolute bioavailability of approximately 50%.
Dyclocaine side effects and Toxicity
Based on the pharmacology of the 5-HT1B/1D agonists, hypertension or other more serious cardiovascular symptoms could occur on overdose.
Dyclocaine Patient Information
No information avaliable
Dyclocaine Organisms Affected
Humans and other mammals
