Dyclonin
Dyclonin Brand names, Dyclonin Analogs
Dyclonin Brand Names Mixture
- No information avaliable
Dyclonin Chemical_Formula
C22H26N2O2S
Dyclonin RX_link
http://www.rxlist.com/cgi/generic3/relpax.htm
Dyclonin fda sheet
Dyclonin msds (material safety sheet)
Dyclonin Synthesis Reference
No information avaliable
Dyclonin Molecular Weight
382.52 g/mol
Dyclonin Melting Point
No information avaliable
Dyclonin H2O Solubility
Readily soluble as hydrobromide formulation
Dyclonin State
Solid
Dyclonin LogP
3.587
Dyclonin Dosage Forms
Tablet for oral administration (24.2 or 48.5 mg)
Dyclonin Indication
For the acute treatment of migraine with or without aura in adults.
Dyclonin Pharmacology
Eletriptan is a selective 5-hydroxytryptamine 1B/1D receptor agonist. In the anesthetized dog, eletriptan has been shown to reduce carotid arterial blood flow, with only a small increase in arterial blood pressure at high doses. While the effect on blood flow was selective for the carotid arterial bed, decreases in coronary artery diameter were observed. Eletriptan has also been shown to inhibit trigeminal nerve activity in the rat.
Dyclonin Absorption
Well absorbed after oral administration with a mean absolute bioavailability of approximately 50%.
Dyclonin side effects and Toxicity
Based on the pharmacology of the 5-HT1B/1D agonists, hypertension or other more serious cardiovascular symptoms could occur on overdose.
Dyclonin Patient Information
No information avaliable
Dyclonin Organisms Affected
Humans and other mammals
