Dyclocainum
Dyclocainum Brand names, Dyclocainum Analogs
Dyclocainum Brand Names Mixture
- No information avaliable
Dyclocainum Chemical_Formula
C22H26N2O2S
Dyclocainum RX_link
http://www.rxlist.com/cgi/generic3/relpax.htm
Dyclocainum fda sheet
Dyclocainum msds (material safety sheet)
Dyclocainum Synthesis Reference
No information avaliable
Dyclocainum Molecular Weight
382.52 g/mol
Dyclocainum Melting Point
No information avaliable
Dyclocainum H2O Solubility
Readily soluble as hydrobromide formulation
Dyclocainum State
Solid
Dyclocainum LogP
3.587
Dyclocainum Dosage Forms
Tablet for oral administration (24.2 or 48.5 mg)
Dyclocainum Indication
For the acute treatment of migraine with or without aura in adults.
Dyclocainum Pharmacology
Eletriptan is a selective 5-hydroxytryptamine 1B/1D receptor agonist. In the anesthetized dog, eletriptan has been shown to reduce carotid arterial blood flow, with only a small increase in arterial blood pressure at high doses. While the effect on blood flow was selective for the carotid arterial bed, decreases in coronary artery diameter were observed. Eletriptan has also been shown to inhibit trigeminal nerve activity in the rat.
Dyclocainum Absorption
Well absorbed after oral administration with a mean absolute bioavailability of approximately 50%.
Dyclocainum side effects and Toxicity
Based on the pharmacology of the 5-HT1B/1D agonists, hypertension or other more serious cardiovascular symptoms could occur on overdose.
Dyclocainum Patient Information
No information avaliable
Dyclocainum Organisms Affected
Humans and other mammals
