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Toprol-XL Marchi, Toprol-XL Analoghi

Toprol-XL Marchi miscela

  • LOPRESSOR HCT
  • Toprol-XL Formula chimica

    C15H25NO3

    Toprol-XL RX link

    http://www.rxlist.com/cgi/generic/metopxl.htm

    Toprol-XL FDA foglio

    Toprol-XL FDA

    Toprol-XL DMS (foglio di materiale di sicurezza)

    Toprol-XL MSDS

    Toprol-XL Sintesi di riferimento

    Brandstorm AE et al. US Pat. 3,873,600 (1975)

    Toprol-XL Peso molecolare

    267.364 g/mol

    Toprol-XL Temperatura di fusione

    120 oC (tartarate salt)

    Toprol-XL H2O Solubilita

    16,9 mg / ml

    Toprol-XL Stato

    Solid

    Toprol-XL LogP

    2.477

    Toprol-XL Forme di dosaggio

    Compressa

    Toprol-XL Indicazione

    Per il trattamento di ipertensione e angina pectoris.

    Toprol-XL Farmacologia

    Metoprololo, un antagonista competitivo adrenergico beta1-selettivo (cardioselettivi), è simile a atenololo nella sua liposolubilità moderata, la mancanza di attività simpaticomimetica intrinseca (ISA), e la membrana debole attività stabilizzante (MSA).

    Toprol-XL Assorbimento

    Rapida e completa, il 50%

    Toprol-XL Tossicita

    LD50 = 5500 mg / kg (per via orale nei ratti), effetti tossici includono bradicardia, ipotensione, broncospasmo e insufficienza cardiaca. LD50 = 2090 mg / kg (per via orale nei topi)

    Toprol-XL Informazioni paziente

    Metoprolol succinate is used to treat high blood pressure alone or in combination with other medications. This medication can also be used to treat a heart condition called angina. This particular formulation is an extended release product, meaning it can be taken once a day. This medication should be taken as directed, with a meal or right after a meal. The tablets should not be broken or crushed. Do not take a double dose if a dose is missed. This medication should not be stopped abruptly; it should be discontinued slowly over time. If you are taking this medication for high blood pressure, make sure to have your blood pressure checked regularly. If you ever have trouble breathing, call your physician immediately. The most common adverse effects are dizziness and tiredness. It is important to inform all your healthcare providers that you are taking this medication, especially before any surgeries or procedures.

    Toprol-XL Atto interessato organismi

    Gli esseri umani e altri mammiferi